abstract |
The present invention relates to the ligands of the A3 receptor of adenosine represented by the general formula (I), their antiagonists, salts, solvates, N-oxides and isomers. IT CONCERNS THE PHARMACEUTICAL COMPOSITIONS CONTAINING THE COMPOUNDS OF THE GENERAL FORMULA (I), THEIR SALTS, SOLVATES, N-OXIDES AND ISOMERS, ON THE USE OF THE COMPOUNDS OF THE GENERAL FORMULA (I), THEIR SALTS, SOLVATES, N-OXIDES AND ISOMERS, ON THE PREPARATION OF THE COMPOUNDS OF THE GENERAL FORMULA (I), THEIR SALTS, SOLVATES, N-OXIDES AND ISOMERS, AND ON THE NEW INTERMEDIATES OF GENERAL FORMULAS (II), (VI), (XI), (XII AND (XV), AND ON THEIR PREPARATION. |