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filingDate 2019-12-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cb9595de0a3d204d5a2d99f3da6d23ad
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6f1489af5fa7a51ac3d757b3c1ae2563
publicationDate 2021-09-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20210117275-A
titleOfInvention saponin conjugate
abstract The present invention relates to an effector moiety capable of inducing an intracellular effect when present inside a mammalian cell, the effector moiety comprising a payload conjugated with one or more saponins. The present invention also relates to an antibody-drug conjugate comprising an effector moiety according to the present invention, or to a ligand-drug conjugate comprising an effector moiety of the present invention comprising an effector moiety comprising a covalently linked saponin. The present invention relates to therapeutic combinations comprising (a) an effector moiety of the invention comprising one or more saponins, and optionally a pharmaceutically acceptable excipient; and (b) an antibody-drug conjugate or ligand-drug conjugate, and optionally a pharmaceutically acceptable excipient. The invention further relates to a pharmaceutical composition comprising an effector moiety of the invention or an antibody-drug conjugate of the invention or a ligand-drug conjugate of the invention, wherein at least one saponin covalently linked to an effector molecule, and optionally pharmaceutically acceptable excipients. The present invention also relates to an effector moiety of the present invention or an antibody-drug conjugate of the present invention or a therapeutic combination of the present invention or a ligand-drug conjugate of the present invention or a pharmaceutical composition of the present invention for use as a medicament. Finally, the present invention also relates to an effector moiety of the present invention or an antibody-drug conjugate of the present invention or a therapeutic combination of the present invention or a ligand-drug conjugate of the present invention for use in the treatment or prophylaxis of cancer or an autoimmune disease or The present invention relates to a pharmaceutical composition.
priorityDate 2018-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID102724971
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92N62
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JVC2
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VKQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63548
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0TWU0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28809
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID439746
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28819
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID225642
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID2158
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7JPZ4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28746
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47958
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5ITF9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP63543
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0UKF2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504969
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28747
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38121
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47966
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419519044
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5P0Z7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ32BG2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IEY2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID373666
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3Q9C9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7IIS0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6TL10
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP11052
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3IKN5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5IZD7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426133118
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VRB8
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25712
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28MD3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47952
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9IQ90
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3B250
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25704
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47956
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0JV33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB3Q9D3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47957
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9IL50
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VAL5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100136560
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0KKD3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7ZWM4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID485430
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91757851
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4LIX2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AYP0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO95832
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2907
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0KAK7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9K8S7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7J0M3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7V7D8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3BSE4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0SIB4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0RFB2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4XU70
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9RFQ2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5GSL0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280800
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4L8U7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0AIX3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5N1Z2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31W50
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9KG97
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08298
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47518
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6SW90
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP30368
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0TNZ8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28319
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ28334
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID3572
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5793
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC6DIG9
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID952
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP47202
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AIK3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3PFJ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7HQG7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0SI58
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7VGF2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4ZUS3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69569
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5I6E1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP08030
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID32821
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1048
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4ZF43
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID374100
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7UR74
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7WKW7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ921I1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0S0M3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3Q0T3
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422154253
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25698
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14254
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5R6D1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92087
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID14255
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M2K2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1043
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6QFH2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92111
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3PNQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A6E4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92112
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3AT37
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5G4S5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0A6E5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9HIQ4
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID17075
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ06435
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71308164
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QQX7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0IFL5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46650
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ZLQ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5M8Z6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5GLQ5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PFK3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7GR20
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46652
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403727
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8KDE0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280705
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7W7H8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1UFB6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP44315
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC4L531
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID11898
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID171101
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7V0X5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31H63
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5QWS1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3NQI1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07750
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID102723407
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419553254
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0KPW6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24337
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ24ZG8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9BM60
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31SC8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7TTW1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ493A5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3815167
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO02837
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA1UZL8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7LHN6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF7CGN2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5CUG9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ92L73
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID280726
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID8617570
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8KA60
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID39824
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6NCS7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7HE42
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0I4M1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449785438
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ49Y73
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5LWG3

Total number of triples: 2117.