http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20210081353-A

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_10a77948035833454698753b762d551a
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-506
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-506
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-14
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00
filingDate 2019-10-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_63201f961f7f63e1a861755dfd917ede
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_207e54fe6262b0ea29af722f856771ca
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a29f9610242f09c41efcacd366bd9c49
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_15abfbaceca85b41d0d0f93b2bd5fb9e
publicationDate 2021-07-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20210081353-A
titleOfInvention Heterocyclic kinase inhibitors and uses thereof
abstract The present invention relates to kinase inhibitors, in particular inhibitors of protein kinases, for example protein-tyrosine kinases LCK, ABL, SRC, KIT, SIK-family and/or mutants thereof. Although structurally similar to dasatinib, the kinase inhibitors of the present invention may exhibit one or more specific properties that distinguish them from dasatinib. The invention also relates to pharmaceutical compositions comprising one or more kinase inhibitors. A kinase inhibitor or pharmaceutical composition of the present invention may be used to treat a disorder or condition, such as a proliferative disorder, such as leukemia or a solid tumor. The kinase inhibitor or pharmaceutical composition may be used in a therapeutic regimen corresponding to, similar to or distinct from that used with dasatinib for the corresponding disorder, in particular one or more additional therapeutic agents, e.g., immuno- It may be used in combination treatment regimens with checkpoint inhibitors.
priorityDate 2018-10-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1140.