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filingDate 2017-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fd27ae9bb6dde762cb0da41870ceb6ef
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publicationDate 2019-06-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20190072565-A
titleOfInvention 1,3-disubstituted cyclobutane or azetidine derivatives as inhibitors of hematopoietic prostaglandin D synthetase
abstract Disclosed are compounds of formula (I) wherein R, R 1 , R 2 , R 3 , Y, Y 1 , a, X and Z are as defined herein. The compounds of the present invention are inhibitors of hematopoietic prostaglandin D synthase (H-PGDS) and may be useful in the treatment of duodenal muscular dystrophy. Accordingly, the present invention further relates to a pharmaceutical composition comprising a compound of the invention. The invention further relates to methods of inhibiting H-PGDS activity and methods of treating disorders associated therewith using a pharmaceutical composition comprising a compound of the invention or a compound of the invention.
priorityDate 2016-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1422.