http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20180026438-A

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filingDate 2016-07-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2ffda8530530077b544f04daa05cf821
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publicationDate 2018-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20180026438-A
titleOfInvention Ethynyl derivatives as metabotropic glutamate receptor modulators
abstract The present invention relates to compounds of the general formula (I), or pharmaceutically acceptable salts or acid addition salts thereof, racemic mixtures, or the corresponding enantiomers and / or optical isomers and / or stereoisomers thereof, (I) In this formula, R &lt; 1 &gt; is lower alkyl; R 2 is phenyl or pyridinyl, wherein the N atom in the pyridinyl group can be in different positions; n is 0, 1 or 2; V and U are independently of each other O or CH 2 , wherein V and U can not be O at the same time; L is a 5 or 6 membered heteroaryl group selected from: . Such compounds may be used for the treatment of Parkinson's disease, anxiety, vomiting, obsessive compulsive disorder, autism, neuroprotection, cancer, depression and type 2 diabetes.
priorityDate 2015-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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