http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20140107574-A

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filingDate 2012-12-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a3e1a0106b8602fa0b53dabf6136a732
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0df5c881aef98a4477533e11982d9520
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publicationDate 2014-09-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20140107574-A
titleOfInvention Compounds for inhibiting the interaction of bcl2 with binding partners
abstract The present invention relates to compounds of formula (I) Compounds of formula I may disrupt BCL-2 interactions with BH3 domain containing proteins. This disturbance of the interaction may restore anti-apoptotic function of BCL-2 in cancer cells and tumor tissues expressing BCL-2. The invention further provides methods of making the compounds of the invention, pharmaceutical formulations comprising such compounds, and methods of using such compounds in the treatment of cancerous diseases. (I) Wherein R 1 , R 2 , R 3 and R 4 are as defined in the description of the invention.
priorityDate 2011-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 794.