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filingDate 2010-02-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7349ea829414967d1686f0aeaeb81a28
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e9a7fd2923c9bdbac3f262bd97957c0e
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publicationDate 2011-10-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20110111313-A
titleOfInvention Isoxazole / O-pyridine derivatives with ethyl and ethynyl linking groups
abstract The present invention relates to novel isoxazole-pyridine derivatives of formula (I) and pharmaceutically acceptable salts and esters thereof. The active compounds of the present invention have affinity and selectivity for GABA A α5 receptors. The invention also relates to a process for the preparation of the active compounds of formula (I), pharmaceutical compositions containing them and their use as medicaments: Formula I Where R 1 , R 2 , R 3 and L are as described herein.
priorityDate 2009-02-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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