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filingDate 2009-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_422216e53deac7a898701db4f5305907
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publicationDate 2010-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20100132180-A
titleOfInvention New Manufacturing Method of Valsartan
abstract The present invention provides a method for preparing valsartan represented by [Formula 1] used as an angiotensin receptor blocker (ARB; also referred to as an angiotensin II receptor antagonist or an AT1 receptor antagonist) as an agent for treating arterial hypertension or heart failure.n n n [Formula 1]n n n n n n n n [Formula 2]n n n n n n n n The method of the present invention is an economical process that is harmless to the human body in only three steps from the intermediate represented by [Formula 2], and is easy and efficient in mass production, and it is possible to synthesize valsartan in high yield and high purity without generating reaction by-products. It is an improved way.
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