http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20080085796-A

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assignee http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_079a5b3eecbeb0e5fcc2e9b817b28c97
classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00
classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K7-06
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07K1-061
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07K7-06
filingDate 2008-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_178480ded155205fee04204df18a9239
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c19f2d0987259675035b6fe276474834
publicationDate 2008-09-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20080085796-A
titleOfInvention Spinorpin derivatives as effective and selective human Ρ2Χ3 receptor antagonists
abstract The present invention relates to spinnor derivatives as effective and selective human P2X 3 receptor antagonists. More specifically, it relates to spinorphine derivatives as effective and selective human P2X 3 receptor antagonists selected from peptide AVVYPWT, peptide LAVYPWT, peptide LVAYPWT, peptide LVVAPWT and peptide cyclic LVVYPWT. The invention also RY gen crispus to Nord to characterize the channel blocking activity and a short recognition of the pin (Xenopus) I recombinant human P2X 3 7 gae alanine scanned RY Nord pin peptide derivative of the receptor expression in the cells of the P2X 3 receptor By measuring the electrophysiological evaluation of cleaved peptide analogs, cyclic peptides and retro-inverso peptides, a novel spinorphine derivative was developed.
priorityDate 2008-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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