http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20070114660-A

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filingDate 2007-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_07327c33ce52dc8564b122a8c1039f53
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publicationDate 2007-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20070114660-A
titleOfInvention ピ lk1-based protein chip, ultra-fast screening method of anticancer substance using the same and anticancer substance obtained by the method
abstract The present invention relates to a Plk1-based protein chip, a high throughput screening method of an anticancer substance using the same, and an anticancer substance obtained by the method. More specifically, Plk1 (polo-like kinase) is a carcinogenic protein on a substrate. Protein chip for detecting interaction between Plk1 substrate protein and PBD, wherein the substrate protein of 1) or PBD (polo-box domain), which is a substrate protein binding site of Plk1, is immobilized, between the PBD of Plk1 and the substrate protein on the protein chip The present invention relates to a method for screening an anticancer substance and an anticancer substance screened by the method, wherein the candidate substance for inhibiting binding is selected as an anticancer substance.n n n The ultrafast screening method of anticancer substances in protein chips according to the present invention can be screened in large quantities quickly and conveniently for binding inhibitors between proteins, including protein interactions, and thus may be usefully used for discovering new anticancer agents.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-9377462-B2
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2012144861-A3
priorityDate 2006-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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