http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20070020400-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4427
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-98
classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4412
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-98
filingDate 2004-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2007-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20070020400-A
titleOfInvention Novel 5,6-dihydropyridin-2-one compounds useful as thrombin inhibitors
abstract There is provided a compound of formula I:n n n n n n n n Wherein R 1 , R 2a , R 2b , R 3a , R 3b , R 4 , R 5 , R 6 , A, G and L have the meanings given in the detailed description.n n n Since the compounds are useful as competitive inhibitors of trypsin-like proteases, such as thrombin and also as prodrugs thereof, they are particularly useful in the treatment of symptoms where inhibition of thrombin is beneficial (e.g. related to thrombo metabolism requiring inhibition of thrombin) Symptoms, and / or diseases in which anticoagulant therapy is needed.
priorityDate 2003-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 481.