http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-20010032687-A

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filingDate 1998-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2001-04-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-20010032687-A
titleOfInvention Conjugates useful in the treatment of prostate cancer
abstract Described herein are chemical conjugates comprising an oligopeptide having an amino acid sequence that is selectively and proteolytically cleaved by a free prostate specific antigen (PSA) and a known cytotoxic agent. The conjugates of the invention are characterized in that the cleavable oligopeptide is attached to an oxygen atom at the 4-position on the deacetylated vinca drug. Such conjugates are useful for treating prostate cancer and benign prostatic hyperplasia (BPH).
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/US-7842581-B2
priorityDate 1997-12-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457810462
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422057620
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID20944
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID152743293
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID440015
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6971259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53975367
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID64335
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25048

Total number of triples: 322.