http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-19990085365-A

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filingDate 1998-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 1999-12-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-19990085365-A
titleOfInvention Biodegradable polymer microspheres capable of continuously controlled controlled release and preparation method thereof
abstract The present invention relates to a microsphere made of a biodegradable polyester-based polymer capable of continuously controlling drug release and increasing the amount of drug encapsulated in the microsphere and a method for preparing the same, which is a drug in a biodegradable polyester-based polymer carrier. By encapsulating the biodegradable polyester-based polymer and the drug through covalent bonding, the drug release rate can be controlled according to the decomposition rate of the biodegradable polyester-based polymer regardless of the diffusion concentration of the drug. As well as to obtain the effect of encapsulating a larger amount of hydrophilic drug in the same size microspheres, the covalent bond of the biodegradable polyester-based polymer and the drug is to preactivate the drug having a functional group and the polymer To the polymer, coupling agents, bases, linkers, spacers Or by adding a multiligand compound to preactivate the polymer and then binding the desired drug.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-100441904-B1
priorityDate 1998-05-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 644.