http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-102348325-B1

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-00
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filingDate 2015-12-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2022-01-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-01-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-102348325-B1
titleOfInvention Anticancer compositions
abstract The present invention relates to androgen receptor (AR)-related diseases or conditions, particularly cancer, more particularly castration-resistant prostate cancer, metastatic castration-resistant prostate cancer, chemotherapy-naive metastatic castration-resistant prostate cancer, biochemically relapsed hormone-sensitive prostate cancer To a pharmaceutical formulation of ARN-509, which may be administered to a mammal, particularly a human, suffering from prostate cancer, including but not limited to, high-risk non-metastatic castration-resistant prostate cancer. In one aspect, this formulation comprises a solid dispersion of ARN-509 and a poly(meth)acrylate copolymer. In one aspect, the solid dispersion of ARN-509 and poly(meth)acrylate copolymer is melt extruded from a mixture comprising ARN-509 and poly(meth)acrylate copolymer, and optionally subsequently melt extruded. It can be obtained by milling the mixture, in particular it is obtained. In one aspect, a solid dispersion of ARN-509 and poly(meth)acrylate copolymer may be obtained by spray drying a mixture comprising ARN-509 and poly(meth)acrylate copolymer in a suitable solvent, in particular is obtained
priorityDate 2014-12-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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