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filingDate 2014-02-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-12-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-102185311-B1
titleOfInvention A site specific conjugate of insulin
abstract In the present invention, the non-peptide polymer and the immunoglobulin Fc region are site-selectively linked to the amino acid residues of the region other than the N-terminus of the insulin beta chain by covalent bonds, thereby enhancing the binding ability with the insulin receptor and thus increasing the activity It relates to an insulin conjugate, a long-acting preparation comprising the same, and a method for preparing the same. The insulin conjugate of the present invention can provide an insulin preparation having significantly increased in vivo activity of a peptide.
priorityDate 2013-02-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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