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filingDate 2019-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2020-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-102170422-B1
titleOfInvention A Novel Tofacitinib Salt, Preparation Methods thereof and Pharmaceutical Compositions Comprising thereof
abstract The present invention relates to tofacitinib camphorsulfonate monohydrate, a method for preparing the same, and a pharmaceutical composition comprising the same. Tofacitinib camphorsulfonic acid salt monohydrate according to the present invention has an equal or higher effect in terms of acceleration, stability under severe storage conditions, photostability, thermal stability, stability according to pH, solubility, etc. as a result of comparison with tofacitinib citrate. Therefore, the pharmaceutical composition of the present invention can be usefully used for preventing or treating diseases selected from the group consisting of rheumatoid arthritis, psoriatic arthritis, and ulcerative colitis.
priorityDate 2018-01-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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