Predicate |
Object |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-07 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J2231-543 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D263-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D205-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J31-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J23-462 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J31-2278 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C251-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-397 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/B01J31-146 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/B01J31-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/B01J23-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D205-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-397 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C251-24 |
filingDate |
2018-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate |
2020-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate |
2020-02-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
KR-102078158-B1 |
titleOfInvention |
Process for preparing Ezetimibe and intermediate thereof |
abstract |
The present invention provides a method for preparing ezetimibe and an intermediate thereof, including a cross-substitution reaction using a second generation Grubbs catalyst and a deprotection reaction using a Perman catalyst. The method for producing ezetimibe of the present invention can be usefully used as an efficient ezetimibe synthesis technique in the pharmaceutical field using ezetimibe as a raw material. |
priorityDate |
2018-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |