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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-519
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filingDate 2015-10-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-101978899-B1
titleOfInvention Novel Pyridopyrimidinone Compounds for Modulating the Catalytic Activity of Histone Lysine Demethylases (KDMs)
abstract The present invention provides a compound of formula (I), a pharmaceutical composition thereof, a process for the preparation of said compound, and a use of said compound as a therapeutic agent, which can modulate the activity of histone lysine demethylating enzyme (KDM). The compounds of formula I act as KDM inhibitors with significant efficacy and have the potential for pharmaceutical intervention of any other disease associated with cancer and KDM control disorders. &Lt; Structural Formula (I) >
priorityDate 2014-10-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424399975
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID78953
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10422
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393374
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419537854
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419584407
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Total number of triples: 689.