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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C231-02
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C231-02
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C233-47
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C231-22
filingDate 2016-01-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2019-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-03-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-101961897-B1
titleOfInvention Preparation method of sacylitol
abstract The present invention relates to a process for the production of Sacubitril (AHU-377, I), one of the components of the new blood pressure lowering drug, LCZ696, which comprises the asymmetric induction reagent (S) -1- ) Cyclic addition, debenzylation, cyclization, esterification and amidation of 2-methyl-2-naphthalenol and 2R-methyl-4-oxo-butanoic acid ). The above production method is easy to obtain the raw material, simple in process, economical and environment-friendly, and is very suitable for industrial production.
priorityDate 2015-01-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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