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filingDate 2009-08-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2016-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-101630217-B1
titleOfInvention [4-(5-Aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-[7-fluoro-1-(2-methoxy-ethyl)-4-trifluoromethoxy-1H-indol-3-yl]-methanone as an inhibitor of mast cell tryptase
abstract The present invention relates to indolbenzylamine compounds useful as inhibitors of tryptamase. The invention also relates to the use of a compound for treating a patient suffering from or susceptible to a physiological condition requiring improvement by inhibition of a tryptase, comprising administering a therapeutically effective amount of the compound to the patient. Furthermore, the present invention relates to a pharmaceutical composition comprising a pharmaceutically effective amount of a compound of formula I, and a pharmaceutically acceptable carrier. Formula I
priorityDate 2008-08-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2734379
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID83717
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452333222
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9955175
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419514433
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408499458
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24323
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID46175649
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID444036
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID452908992
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6V115
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822168
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1117
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281068
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119440
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID237940
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID46175648
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449282311
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453612601
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419589583
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID412584818
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID411555350
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453831981
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448301204
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3776
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID66111
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119236
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453739895
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18362537
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21925356

Total number of triples: 337.