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filingDate 2006-09-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2012-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2012-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber KR-101214433-B1
titleOfInvention Condensed heterocyclic derivatives, pharmaceutical compositions containing the same and uses thereof
abstract The present invention is expressed by the following general formula (I), which expresses human SGLT activity inhibitory activity and is useful as a prophylactic or therapeutic agent for diseases caused by hyperglycemia, such as diabetes, postprandial hyperglycemia, abnormal glucose tolerance, diabetic complications, obesity, and the like. Nitrogen-containing condensed ring derivatives or pharmacologically acceptable salts thereof, or prodrugs thereofn n n (R 1 and R 4 are either one of the groups represented by general formula (S) (R 5 and R 6 are H, OH, a halogen atom, etc .; Q is an alkylene group; ring A is an aryl group, etc.), the other Side is H, OH, an amino group, etc .; R 2 and R 3 are H, OH, an amino group, a halogen atom, a substitutable alkyl, and the like; A 1 is O, S, or the like; A 2 is CH, or N; G is a group represented by the following general formula (G-1) or (G-2) (E 1 is H, F or OH; E 2 is H, F, methyl group, etc.), and a pharmaceutical composition containing the same and its It is to provide a medical use.n n n SGLT activity inhibitory effect, hyperglycemia, condensed heterocyclic derivative
priorityDate 2004-03-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA7H492
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421061784
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68718338
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1PM04
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415740930
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID12918
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67515
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6438331
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1175
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18530292
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64560
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450396029
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532926
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID34152
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ93MW7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID656629
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424506096
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35576
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ93IM5
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID21758144
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100150233
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ09541
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB7NPS4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559505
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID72006
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43428
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410831523
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81881
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3921488
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5PNF2
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5282210
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID409979

Total number of triples: 1305.