http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-100882972-B1
Outgoing Links
| Predicate | Object |
|---|---|
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D285-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C323-63 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C12P41-005 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C323-59 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C12P13-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C12P11-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C323-63 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C323-59 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C12P41-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C12P13-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C12P17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D285-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C12P11-00 |
| filingDate | 2002-09-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2009-02-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 2009-02-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | KR-100882972-B1 |
| titleOfInvention | Enzymatic Methods for Preparation of Substituted 2-Amino-3- (2-Amino-phenylsulfanyl) -propionic Acid |
| abstract | The compounds of formula (I) are useful for the preparation of 1,5-benzothiazepines useful as enzyme inhibitors such as proteases, interleukin-1β-converting enzymes, elastase or angiotensin enzymes, GPCR antagonists (cholescystokinin, angiotensin II receptor). The present invention relates to a novel process for preparing a compound of formula (I) comprising reacting a compound of formula (II) with a protease in an aqueous system containing an organic co-solvent:n n n Formula In n n n n n n n Formula IIn n n n n n n n Wheren n n R 1 , R 2 , R 3 , n and R 4 are as described in the specification. |
| priorityDate | 2001-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
| Predicate | Subject |
|---|---|
| isDiscussedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10222027 http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426445153 |
Total number of triples: 23.