http://rdf.ncbi.nlm.nih.gov/pubchem/patent/KR-100461569-B1
Outgoing Links
Predicate | Object |
---|---|
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-04 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-04 |
filingDate | 2002-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 2004-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 2004-12-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | KR-100461569-B1 |
titleOfInvention | Process for producing optically pure 3-hydroxy-pyrrolidine |
abstract | The present invention relates to a method for preparing optically pure 3-hydroxy-pyrrolidine, and more particularly, to react with ammonia and an aldehyde compound using 3,4-epoxy-1-butanol having optical activity as a starting material. After preparing the 4-protected imino-butane-1,3-diol, the hydroxy group at the C-1 position is selectively activated, or subsequently treated with an acid to convert the imino group into an amine group, and then in the presence of a base. By carrying out an intramolecular cyclization reaction, it relates to a novel process for producing 3-hydroxy-pyrrolidine represented by the following formula (1) economically and simply in high yield optically.n n n n n n n n n n In Chemical Formula 1, * represents a compound (S) or (R) having optical activity. |
priorityDate | 2002-05-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 67.