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filingDate 2013-09-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2016-08-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-WO2014034929-A1
titleOfInvention Oral sustained release pharmaceutical composition containing hydromorphone hydrochloride
abstract Sustained-release pharmaceutical for oral administration containing hydromorphone hydrochloride or oxycodone hydrochloride hydrate, which exhibits reliable main pharmacological effects and has excellent formulation stability that avoids excessive release of main agents such as alcohol tolerance The challenge is to provide a composition. (A) Hydromorphone hydrochloride or oxycodone hydrochloride hydrate, (B) hydroxypropylmethylcellulose acetate succinate having a median diameter (D 50 ) of 40 μm or less, (C) hydroxypropylcellulose, and (D) a saccharide , The sustained release pharmaceutical composition, wherein the weight ratio (C) / (B) of the component (B) to the component (C) in the composition is 11/3 to 3/11.
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