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filingDate 2010-02-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2012-09-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-WO2010098344-A1
titleOfInvention Tricyclic pyrazolopyrimidine derivatives
abstract To provide a novel compound that inhibits the action of HSP90, particularly a novel compound that inhibits the function of HSP90 as a chaperone protein and has antitumor activity. The present invention relates to a pyrazolopyrimidine compound represented by formula (1) having various substituents, which inhibits the ATPase activity of HSP90 and has antitumor activity, and an HSP90 inhibitor comprising a compound represented by formula (1) , A pharmaceutical comprising the compound represented by formula (1), an anticancer agent comprising the compound represented by formula (1), a pharmaceutical composition comprising the compound represented by formula (1) and the formula (1) A method for treating cancer using the compound is provided.
priorityDate 2009-02-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 401.