Predicate |
Object |
classificationCPCAdditional |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y10T428-13 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y10T428-2982 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-1623 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-1652 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-0075 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K38-00 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-454 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-19 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-24 |
filingDate |
2006-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate |
2008-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
JP-WO2006095788-A1 |
titleOfInvention |
Particles and formulations containing the particles |
abstract |
The present invention relates to tert-butyl (4R) -4-{[((1R) -2-[(1-benzylpiperidin-4-yl) amino] -1-{[(cyclohexylmethyl) thio] methyl} -2. -Oxoethyl) amino] carbonyl} -1,3-thiazolidine-3-carboxylate containing particles having an average particle diameter of 0.01 to 20 [mu] m. Since the preparation containing the particles has excellent ability to migrate to the lungs by inhalation and is excellent in dispersibility as particles, it is easy to handle, and the compound can be used as a transpulmonary preparation. |
priorityDate |
2005-03-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |