http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-S54106466-A
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_e7962109cd4763907b82b66760cd0ae8 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D285-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D261-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-56 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-54 |
filingDate | 1978-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e4a7685fa08d060d9f937acad819c99a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_af875d0930b208ac2025f14d72722048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_41772e0b9227175e5ab1fc1df660fad6 |
publicationDate | 1979-08-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | JP-S54106466-A |
titleOfInvention | Preparation of heterocyclic compound |
abstract | PURPOSE: To prepare a heterocyclic compound useful as an intermediate for medicines and pesticides, in high yield in a simple operation advantageously, by reacting safe and easily handleable acyl Medlrm's acid or its homolog with an amino compound. n CONSTITUTION: An acyl derivative of Meldrums acid of formula I: (R 1 , R 2 , and R 3 are lower alkyl groups) or its homolog is reacted with a compound of formula II: (R 4 is H, alkyl, or (un)substituted phenyl group; X is -CO-,-CS-, or -SO 2 -), hydroxylamine (hydrochloride, sulfate, etc.) or a hydrazine of the formula R 5 NH NH 2 (R 5 is the same as R 4 ) under heating or melting, and, if necessary, in an inert solvent, at room temperature to refluxing one to give a hetercyclic compound consisting of a compound of formula III, an isoxazole derivative of formula IV, or a pyrazole derivative of formula V. The raw material can be readily obtained by acylating Meldrum's acid according to the conventional method. n COPYRIGHT: (C)1979,JPO&Japio |
priorityDate | 1978-02-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 30.