abstract |
(57) [Summary] The present invention has vasopressin antagonism and the like, and has the general formula (I): [Wherein, R 1 is aryl or the like which may be substituted with lower alkoxy, R 2 is lower alkyl or the like, R 3 is hydrogen or the like, R 4 is lower alkoxy or the like, R 5 Is hydrogen or the like, A is NH or the like, E is -C (= O)-or the like, X is -CH = CH-, -CH = N- or S, and Y is CH or N The present invention relates to a novel benzamide derivative represented by the formula: |