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filingDate 1996-01-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 1998-11-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-H10512245-A
titleOfInvention Compositions and methods for transdermal delivery of acid labile drugs
abstract (57) [Summary]nA composition for reducing acid instability of a transdermal penetration enhancing drug and related methods are described. (A) a therapeutically effective amount of a pharmacologically active drug susceptible to acid-catalyzed degradation; (b) a pharmaceutically acceptable carrier substantially free of lower alkanols; and (c) penetration of functional derivatives of fatty acids. A transdermal composition comprising an enhancing amount. Such compositions increase the utility of transdermal compositions that rely on organic acids, such as oleic acid penetration enhancers.
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