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filingDate 1994-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 1997-04-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-H09503492-A
titleOfInvention Succinamide derivatives, their preparation and their use as gelatinase and collagenase inhibitors
abstract (57) [Summary] A compound represented by the formula (1) (in the formula, R 1 represents (a), R 3 represents a hydrogen or halogen atom, a methyl, trifluoromethyl or methoxy group, and R 2 represents a hydrogen atom. Or a methyl group) and its salts, solvates, hydrates, and prodrugs. The compounds are potent and selective metalloproteinases, long-acting, orally active inhibitors of gelatinases, which in particular inhibit angiogenesis in vivo. Therefore, they can be expected to be used for the prevention or treatment of angiogenesis-dependent diseases such as solid tumors and arthritis diseases.
priorityDate 1993-08-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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