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filingDate 1992-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 1993-10-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-H05255116-A
titleOfInvention Pharmaceutical formulations for oral administration
abstract (57) [Summary] (Modified) [Objective] To provide a pharmaceutical preparation suitable for oral administration, which comprises a pharmaceutically useful methanediphosphonic acid derivative. [Structure] Adjuvant containing a pharmaceutically useful methanediphosphonic acid derivative represented by the general formula I as an active ingredient and a macromolecular cyclic polyether represented by the general formula (II) as an absorption enhancer, and being pharmaceutically acceptable A pharmaceutical preparation which is effective for the treatment of hypercalcemia and osteolytic bone metastasis, which contains [In the formula (I), R 1 and R 2 are halogens, one of them is H and the other is phenylthio group, cycloalkylamino group, or the like, or one of them is H and OH and the other is alkyl. , (Mono (di) substituted) aminoalkylene, (Phenyl-substituted) alkyleneaminoalkylene groups and the like. In the formula (II), X 1 to X 4 are -COOH,- CONH 2 etc.]
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2011508757-A
priorityDate 1991-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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