http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-H04253973-A
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_5dfc0b033ac4c841466d97a5f28ea32b |
classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P31-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-435 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 |
filingDate | 1991-04-19-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8ec7800d6ccc9a18ff8fe3a1de2af4b1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a231c143931ea740b35cadf67a06bce1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_36110d3dd9c00ad88cb87f5bea5c3775 |
publicationDate | 1992-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | JP-H04253973-A |
titleOfInvention | Pyridonecarboxylic acid derivative |
abstract | PURPOSE: To provide a new compound having strong antibacterial activity against sensitive and resistant Gram-positive and Gram-negative bacteria and useful for the treatment of bacterial infectious diseases. n CONSTITUTION: The compound of formula I [R 1 is lower alkyl or phenyl; R 2 and R 3 are H or lower alkyl; R 4 is H, etc. ; X is N or C-Y (Y is H, halogen, etc.); m and n are 0 or 1; the dotted line is single or double bond], e.g. 7-[(1R*,2 R*,6S*)-2-amino-8-azebicyclo[4,3,0]non-3-en-8-yl]-1-cyclopropyl-6,8-difluoro-1,4- dihydro-4-oxo-3-quinolinecarboxylic acid. The compound can be produced by reacting a compound of formula II [R 7 is H or carboxyl-protecting group; R 40 is H, etc.; X is N or C-Y (Y is H, halogen, etc.); Z is eliminable group] with a compound of formula III (R 20 and R 30 are H, amino-protecting group or lower alkyl; m and n are 0 or 1) and, as necessary, removing the protecting group from the resultant compound of formula IV. n COPYRIGHT: (C)1992,JPO&Japio |
isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0705828-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0704443-A2 |
priorityDate | 1990-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 24.