http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-5437525-B1
Outgoing Links
Predicate | Object |
---|---|
classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/Y02P20-55 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C271-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C227-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C229-36 |
classificationIPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B57-00 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C303-30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C269-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07F7-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C271-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C309-73 |
filingDate | 2013-09-27-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 2014-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 2014-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | JP-5437525-B1 |
titleOfInvention | Tyrosine derivative and method for producing tyrosine derivative |
abstract | In addition to tyrosine derivatives useful as melatonin MT 1 receptor antagonists, the present invention introduces an iodo group with good regioselectivity and high yield at the para-position of the phenolic hydroxyl group in the benzene ring of m-tyrosine. And it aims at providing the method of manufacturing a specific m-tyrosine derivative efficiently. A tyrosine derivative according to the present invention is represented by the following formula (I). [Wherein R 1 represents an amino-protecting group, etc .; R 2 represents a carboxy-protecting group, etc .; R 3 represents a hydrogen atom group, etc .; R 4 represents a halogen atom group, etc .; , — (CH 2 ) 1 — [Z (CH 2 ) m ] n —; X represents a leaving group] [Selection figure] None |
isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014103998-A3 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-2894476-A1 |
priorityDate | 2012-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 126.