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filingDate 2020-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2023-02-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2023504038-A
titleOfInvention Formulations of ion channel modulators and methods of preparation and use of ion channel modulators
abstract The present invention relates, in part, to fused heteroaryl compounds useful for preventing and/or treating diseases or conditions associated with abnormal functioning of voltage-gated sodium ion channels, e.g., abnormal protracted/protracted sodium currents. of composition or dosage form comprising Neurological disorders (e.g., Dravet syndrome, epilepsy), pain, neuromuscular disorders, trigeminal-autonomic headache (TAC), migraine, cranial neuropathy or polyneuropathy, and cortical spreading depression (CSD) Also provided herein are methods of treating diseases or conditions associated with abnormal function of sodium ion channels, including: In another aspect, the invention provides a method of making an ion channel modulator.
priorityDate 2019-11-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2764
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID146570
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60880
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2763
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID38103
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81423
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2160
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504036
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MHY7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5RDS9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID407490353
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID60444
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID9541
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2405
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504078
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3821
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419493319
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2754
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01315
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503865
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00749
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP96471
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP81025
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154496482
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID110876
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44383
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423390420
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154496480
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5282474
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5486971
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6741
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448532098
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503925
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535975
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503920
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67968
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419479210
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9YHC5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID433322164
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67970
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID443872
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422601179
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503133
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67973
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01334
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67971
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451339314
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01331
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419538410
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419578152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449148440
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01336
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID41375
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419578149
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP67974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503199
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114690
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01340
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP06869
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2162
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01339
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5282452
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8146
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP01342
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JLN9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2724385
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447893194
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54891
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503083
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60606
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419503121
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID198429
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID54892
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID37768
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536333
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ05589
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491273
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ98TA8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID105421565
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91WL8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426147843
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4170
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559527
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4171
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID449067953
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95LG8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450394443
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419491537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451466641
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP16227
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100004419
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID114781
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448969875
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID44263857
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5281006
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419536232
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5388962
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134543335
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419554785

Total number of triples: 728.