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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/G01N33-57434
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H17-04
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filingDate 2020-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2022520798-A
titleOfInvention Prostate-specific membrane antigen (PSMA) ligand containing a linker capable of cleaving amylase
abstract In particular, the present invention relates to a PSMA binding ligand comprising an oligosaccharide constituent block containing a binding that can be cleaved by alpha-amylase. Typically, this PSMA binding ligand further comprises a PSMA binding motif Q and a chelating agent residue A, wherein the PSMA binding motif Q and the chelating agent residue A preferably contain at least one linker comprising an oligosaccharide constituent block. Linked via AL AQ -Q, the PSMA binding ligand therefore preferably has structure (I) or a pharmaceutically acceptable salt or solvate thereof. [Selection diagram] None
priorityDate 2019-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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