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filingDate 2019-12-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2022514385-A
titleOfInvention 3α-Hydroxy-17β-amide neurostimulatory steroids and their compositions
abstract Equation (I) Compounds of or pharmaceutically acceptable salts thereof are provided herein, R 2a , R 2b , R 4a , R 4b , R 6 , R 7 , R 11a , R 11b , R 16 , R 17 , ,. R 3 , R 5 , R 19 , RX and RY are as defined herein. Also provided herein are pharmaceutical compositions comprising a compound of formula (I) and, for example, methods of using the aforementioned compounds in the treatment of CNS-related disorders. For example, compounds designed to act as GABA regulators are provided herein. In some embodiments, such compounds are envisioned to be useful as therapeutic agents for treating CNS-related disorders.
priorityDate 2018-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID429714538
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID134664
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2760920
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID123042
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457460012
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68156
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456468049
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143026
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID25674
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID67446
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426264270
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419546878
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143011
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453727523
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143102
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7400
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87601
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415810366
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143027
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419523291
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5152094
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415676723
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419485969
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468142036
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID294739
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468142035
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415716027
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153622515
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143513
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143511
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9VV43
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Z2D6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163590756
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143709
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456485498
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143517
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419584807
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456485349
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143381
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID947
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419474462
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143502
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID519935
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID468143486
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414876452
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID37818722
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453346386
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID539629
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ00566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69321
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419507876
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3016
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456366051
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID18096
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6473767
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5493302
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID119
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419577629
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466958334
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393276
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID962
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419474470

Total number of triples: 380.