http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2022513959-A

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filingDate 2019-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-02-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2022513959-A
titleOfInvention Macrocycles and their use in the treatment of diseases
abstract The present invention has the formula (I) capable of regulating the activity of CFTR. [Chemical 1] (In the formula, all variables are as defined herein) with respect to the heterocyclic compound. The present invention further provides a method for producing the compounds of the present invention, and therapeutic uses thereof. The present invention further provides methods of their preparation, their medical use, in particular their use in the treatment and management of diseases or disorders, including cystic fibrosis and related diseases.
priorityDate 2018-12-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ108U0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF6QRS1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68243
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26361
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10439
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447931045
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26362
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP68245
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID19960
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP18109
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163440488
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID408285
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9896267
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26363
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8070
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421442122
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID450473
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465317566
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154963115
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3530572
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420490669
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID154963116
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421916567
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419529444
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419513968
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJI4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419502369
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448551087
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422035037
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3037032
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406935959
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465353579
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ00PJ2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419586450
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457633272
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22379495
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJT9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID431904250
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5333
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425234083
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6918554
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420993972
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID273
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC0HJU0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87207651
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393348
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID423224442
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID421529
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419505573
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID159087
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6809
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID163772067
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24350
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2QL74
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID153618241
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2QL83
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559581
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP42633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2QLA3
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID465386717
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6610344
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4122349
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419532030
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2QLB4
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419483985
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID26954391
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID466039776

Total number of triples: 709.