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filingDate 2020-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2022505053-A
titleOfInvention BTK inhibitors, their pharmaceutically acceptable salts and crystalline polymorphs, and their applications
abstract The present invention provides BTK inhibitors and pharmaceutically acceptable salts thereof, polymorphs thereof and applications thereof. Specifically, the present invention relates to (R) -6-((1-acryloylpiperidin-3-yl) amino) -7-fluoro-4-((2-fluoro-4-morpholinophenyl) amino) -1. , 2-Dihydro-3H-pyrrolo [3,4-c] Pyridine-3-one or a pharmaceutically acceptable salt thereof, a polymorph of crystals and applications thereof. Furthermore, the present invention discloses a pharmaceutical composition containing the inhibitor and its application. [Selection diagram] None
priorityDate 2019-03-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 36.