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filingDate 2019-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2022-01-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2022503942-A
titleOfInvention Isoindoline compounds, methods of preparation thereof, pharmaceutical compositions and uses
abstract The present invention relates to a polysubstituted isoindoline compound represented by the general formula (I), a method for preparing the same, a pharmaceutical composition and an application thereof. Specifically, the polysubstituted isoindoline compound provided in the present invention has stronger antitumor activity and antitumor spectrum as a novel structural CRL4CRBNE3 ubiquitin ligase regulator and treats diseases related to CRL4CRBNE3 ubiquitin ligase. Can be used in the preparation of drugs to be used.
priorityDate 2018-09-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49459
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6646980
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9FMM0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49427
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9FWT2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Y2X8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393636
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6H795
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID80479
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425193155
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XWF6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID38456
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421949246
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID30386
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10352977
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10387
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421183054
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID8113
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393705
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6632727
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID23136949
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2TA10
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9Z255
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414752517
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95044
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95LM1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2T9X7
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6386
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94490
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7054
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2TA03
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ94F47
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9H832
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ93571
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ941B6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457311044
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450645223
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8SWD4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12488879
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP92974
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8AVU2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420657017
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP02248
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID107639
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2775088
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2736069
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415731140
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ91W82
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15187046
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426640850
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO00762
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419557048
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415799373
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457532997
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7ZY08
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425348537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419553602
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP56616
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1RML1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID6536467
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453706522
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7YQJ9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP93028
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID75809
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7Z7E8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13398716
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ921J4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11423623
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID406970473
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ553Y7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419489076
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17973618
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7TSS2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457193495
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF4HPP7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425386533
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419860824
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414662412
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135399369
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15559658
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1RMX2
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414862846
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35135
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426138477
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO00102
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO00103
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID12313776
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35133
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1923
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9845
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCI1RRW0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15187050
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5RF84
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35134
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421058420
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35130
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID977
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35131
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6547
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35128

Total number of triples: 729.