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filingDate 2019-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2021-05-06-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2021511315-A
titleOfInvention Substituted pyrazolo [3,4-d] pyrimidine compounds as RET kinase inhibitors
abstract Provided herein are Formula I: [Chemical 1] Compounds and their tautomers, as well as pharmaceutically acceptable salts and kinases, where R 1 and R 2 have the meanings given herein and these are RET. Kinase inhibitors are useful in the treatment and prevention of diseases that can be treated with RET kinase inhibitors, including diseases and disorders associated with RET.
priorityDate 2018-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822236
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27097
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16542
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5280343
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID24350
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822235
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1576
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10184653
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1749976
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53406297
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID126591927
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822234
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10096
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ58546
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822230
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO77620
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ06PM8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419481666
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451084827
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID822224
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447543134
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID462301
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP35866
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID937623
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424634595
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10765
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID403989
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID77727
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID514062
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419479188
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53315854
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11167602
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9ZKT0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9210
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID28886829
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419478793
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID824497
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419475039
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID28886826
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139336336
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HJ69
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82191
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453757922
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID852825
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP55151
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53358942
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID71255631
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID644241
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0C647
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID824011
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP26724
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID52788
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID408213589
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID823990
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27259
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6442177
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP10618
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID823989
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP27258
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID823987
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419604742
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3MTU1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53235510
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID823986
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425930438
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID542367
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID823985
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID139331013
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419486252
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP55971
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID821554
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID447687512
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID779087
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135539077
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4072
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419592141
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID821461
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID450907777
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416109377
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID4893
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424636277
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3NEV8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46827

Total number of triples: 1695.