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filingDate 2021-05-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_514e74b17b007dac05bde74a0132e296
publicationDate 2021-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2021130673-A
titleOfInvention Pharmaceutical composition containing indole derivative, its preparation method and its use
abstract PROBLEM TO BE SOLVED: To prepare a clear and stable pharmaceutical composition containing an indole derivative, a method for preparing a dihydrochloride containing a high content of a pharmacologically active isomer suitable for industrial production, and a pharmaceutical composition. Provide use of. A lyophilized pharmaceutical composition for use in the treatment of cancer, comprising a pharmacologically active compound of a pharmaceutically acceptable general formula 1a dihydrochloride: In the formula, R is CH 3 , R 1 is 6-CH 3 , R 2 is H; X is N; Y is N, at least 95 of the pharmacologically active compounds. %% by weight (w / w) is in the form of the E isomer. [Selection diagram] None
priorityDate 2015-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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