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filingDate 2018-08-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-11-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2020531540-A
titleOfInvention Sustained-release anesthetic composition and its preparation method
abstract Anesthesia compositions for topical administration of amide-type anesthetics to the subject in need are provided. This anesthetic composition is prepared by hydrating a highly captured lipid structure containing an amide anesthetic and a lipid mixture with an aqueous buffer solution at a pH higher than 5.5, the captured amide anesthetic. It has a multi-layered endoplasmic reticulum with the drug. For large-scale production and for preparing anesthetic compositions using simpler and more viable processes to provide a higher molar ratio of amide anesthetic to phospholipids compared to prior art. Methods are also provided. This anesthetic composition has a long duration of efficacy suitable for drug delivery. [Selection diagram] FIG. 3B
priorityDate 2017-08-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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