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filingDate 2017-12-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-05-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2020515507-A
titleOfInvention Activity-based probe compounds, compositions, and methods of use
abstract Activity-based probe compounds are provided for use in labeling cysteine proteases. These compounds are targeted to proteases via specific targeting elements. These compounds further include a detectable element such as a fluorescent label, a radioactive label or a chelator. In some cases, these compounds further include a quenching element that is released upon reaction with the protease. Also provided are compositions comprising these compounds and methods for using these compounds, eg, in labeling proteases in animals and in visualizing tumors in animals.
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