http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2020506902-A

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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4985
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filingDate 2018-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2020-03-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2020506902-A
titleOfInvention Substituted pyrazolo [1,5-a] pyrazine compounds as RET kinase inhibitors
abstract Compounds of Formula I, and stereoisomers and pharmaceutically acceptable salts or solvates thereof, are provided herein, wherein A, B, D, E, X 1 , X 2 , X 3 , and X 4, RET inhibitors of kinases, have the meaning given herein, including diseases and disorders mediated by RET kinase, diseases that can be treated with RET kinase inhibitor Useful for treatment and prevention. Embedded image
priorityDate 2017-01-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422072509
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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID43875
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419496987
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9XSJ6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426069337
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP58839
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID430153713
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC3NGT6
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11000522
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID427737345
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Total number of triples: 1337.