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publicationDate 2020-05-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2020079249-A
titleOfInvention Pharmaceutical composition of Tecobilimat for injection and method for preparing same
abstract Tecobilimat (4-trifluoromethyl-N-(3,3a,4,4a,5,5a,6,6a-octahydro-1,3-dioxo), a highly active small molecule viral inhibitor -4,6-Ethenocycloprop[f]isoindol-2(1H)-yl)-benzamide), which has improved poor water solubility. SOLUTION: The pharmaceutical composition of tecobilimat (compound of formula 1), cyclodextrin as an active ingredient, cyclodextrin and an additive, wherein said additive is meglumine. . [Selection diagram] None
priorityDate 2016-07-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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