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filingDate 2017-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-12-19-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2019536757-A
titleOfInvention 1,3-Disubstituted cyclobutane or azetidine derivatives as hematopoietic prostaglandin D synthase inhibitors
abstract A compound of formula (I) wherein R, R 1 , R 2 , R 3 , Y, Y 1 , a, X, and Z are as defined herein. The compounds of the present invention are inhibitors of hematopoietic prostaglandin D synthase (H-PGDS) and may be useful in treating Duchenne muscular dystrophy. Thus, the present invention is further directed to a pharmaceutical composition comprising a compound of the present invention. The present invention is further directed to methods of inhibiting H-PGDS activity and treatment of disorders associated therewith using a compound of the invention or a pharmaceutical composition comprising a compound of the invention. [Chemical 1]
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2020530446-A
priorityDate 2016-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 1412.