http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2019507799-A

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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J43-003
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filingDate 2016-12-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2019-03-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2019507799-A
titleOfInvention Steroid compound, composition containing the compound and use thereof
abstract The present invention provides steroidal compounds, compositions comprising such compounds and uses thereof. Specifically, the present invention relates to a steroid compound represented by the formula (I), as well as the compound or a crystal form thereof, a pharmaceutically acceptable salt, hydrate or solvate, stereoisomer, prodrug, Disclosed are pharmaceutical compositions comprising a metabolite or isotopic isomer. The compounds according to the invention are used as CYP17 enzyme inhibitors and have better pharmacokinetic parameter properties, which can improve the drug concentration of the compounds in the body of the animals, whereby the efficacy and safety of the drugs It is used for the preparation of a drug to improve the disease and to treat diseases associated with CYP17 enzyme (eg, prostate cancer etc.).
priorityDate 2016-02-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 504.