http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2019001811-A

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filingDate 2018-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1ac958f4b374962ce6c8afe4dfc1e720
publicationDate 2019-01-10-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2019001811-A
titleOfInvention 2-((R) -2-methylpyrrolidin-2-yl) -1H-benzimidazole-4-carboxamide crystal form 1
abstract 2-((R) -2-methylpyrrolidin-2-yl) -1H-, which is a poly (ADP-ribose) polymerase (PARP) inhibitor and is also referred to as ABT-888, which is easy to produce and prepare. Provided are benzimidazole-4-carboxamide crystal form 1, a production method thereof, a composition containing the same and a production method using the same, and a method for treating a patient having a disease using the same. When measured at about −100 ° C. in a square crystal system and a P43212 space group with radiation at 0.7107 個 々, the individual lattice parameter values a, b and c are 8.218 Å ± 0.002 Å, 8 2-((R) -2-methylpyrrolidin-2-yl) -1H-benzimidazole having 218Å ± 0.002Å and 36.06Å ± 0.01Å and α, β and γ values of 90 ° 4-Carboxamide crystal form 1. [Selection figure] None
priorityDate 2007-10-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 618.