http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2018518489-A

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classificationCPCAdditional http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07B2200-13
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classificationCPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D209-48
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C315-06
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C315-04
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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C317-28
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filingDate 2016-06-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-07-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018518489-A
titleOfInvention Preparation method of apremilast and its intermediate
abstract The present invention relates to a process for the preparation of 1- (3-ethoxy-4-methoxy-phenyl) -2-methanesulfonyl-ethylamine of formula (II), its resolution and its use in the preparation of apremilast of formula (I), Process for the preparation of crystalline form B, an amorphous form of apremilast and a process for preparing a crystalline form of (S) -1- (3-ethoxy-4-methoxy-phenyl) -2-methanesulfonyl-ethylamine of formula (Va) . [Selection] Figure 2
priorityDate 2015-06-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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