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filingDate 2016-05-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2018-06-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2018515593-A
titleOfInvention Pyrazolo [4,3-c] quinoline derivatives for the inhibition of β-glucuronidase
abstract The present invention provides a novel pyrazolo [4,3-c] quinoline derivative exhibiting specific inhibitory activity against microbial β-glucuronidase, and is a potent agent for preventing chemotherapy-induced diarrhea (CID) in cancer. Provides activity. Thus, the compounds of the present invention (1) prevent chemotherapy-induced diarrhea (CID), enhance chemotherapy chemotherapy efficiency, and (2) prevent carcinogens from causing colon cancer. For health food supplements. [Selection] Figure 1
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO60656
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP36537
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID91666371
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458393636
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7400
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID124093769
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457653144
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID124093784
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414144546
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HAW8
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9321
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6327614
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ64550
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3SY77
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HAW7
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415133005
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8JZZ0
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ3UP75
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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6PDD0
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3397
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID417081947
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Total number of triples: 419.